Ionic Strength Dependency Analysis evaluates how the solubility and stability of a drug substance are influenced by the concentration of ions (e.g., salts, buffers) in a solution. This test is critical for optimizing formulations intended for physiological fluids (e.g., blood, gastrointestinal fluids) and ensuring compliance with USP <1151> and ICH Q6A guidelines.
Ionic strength quantifies the total concentration of ions in a solution and is calculated as:
Ionic Strength Dependency Analysis measures how changes in Ionic Strength (via added salts, buffers, or counterions) affect:
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Drug solubility: Salts can increase (salting-in) or decrease (salting-out) solubility.
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Colloidal stability: Ionic strength impacts zeta potential and aggregation in nanosuspensions.
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Protein conformation: High II may destabilize biologics via charge shielding or Hofmeister effects.
Fig.1 Effect of ionic strength on the solubility of a specific protein in NaCl solution. (STEMart Original)
Key Test Parameters
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Solubility vs. Ionic Strength: Measure solubility in NaCl, KCl, or buffer solutions across different ionic strengths.
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Critical Coagulation Concentration (CCC): Determine the ionic strength at which colloids aggregate (via DLS or turbidity).
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pH-Ionic Strength Interplay: Assess combined effects of pH and ionic strength on ionization and solubility.
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Excipient Compatibility: Test common buffers for salting-out risks.
Measurement Technologies
Shake-Flask Method (USP <1176>)
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Principle: Saturate drug in solutions of varying ionic strength, filter, and quantify dissolved API.
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Results: Solubility vs. ionic strength curves.
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High accuracy for thermodynamic solubility.
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Compatible with HPLC/UV-Vis quantification.
Potentiometric Titration
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Principle: Use ion-selective electrodes to measure activity coefficients and calculate II effects.
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Results: Activity vs. ionic strength profiles.
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Direct measurement of ion-drug interactions.
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Automated systems (e.g., Sirius T3) enable high-throughput screening.
Dynamic Light Scattering (DLS)
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Principle: Monitor particle size changes as ionic strength increases to detect aggregation.
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Results: Hydrodynamic diameter and CCC values.
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Real-time tracking of colloidal instability.
Zeta Potential Analysis
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Principle: Measure surface charge (zeta potential) to predict electrostatic stabilization.
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Results: Zeta potential vs. ionic strengths plots.
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Identifies critical II thresholds for colloidal systems.
Partner With Us
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Holistic Expertise: From ionic strength screening to formulation mitigation.
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Advanced Tools: Sirius T3, Malvern Zetasizer, and HPLC-MS for ion-drug interaction studies.
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Regulatory Alignment: Protocols pre-validated for FDA/EMA submissions.
For more information on our Ionic Strength Dependency Analysis service or to discuss your specific requirements, please contact us today.